SCHEMBL8429205

SCHEMBL8429205

CC(C)(C)CC(=O)N(N)C(Cc1ccccc1C(=O)c1cc(NC=NN)cc(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.34
BCHE P06276 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.32
KCNA5 P22460 1/20 0.31
PPARG P37231 1/20 0.31
ALDH1A1 P00352 1/20 0.30
KDM4E B2RXH2 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428874 0.91 BCHE (0.34) TACR1BCHETAS2R14KCNA5ALDH1A1
SCHEMBL8432545 0.85 BCHE (0.32) TACR1BCHETAS2R14KDM4ESMN1; SMN2
SCHEMBL8429100 0.83 BCHE (0.34) TACR1BCHETAS2R14KCNA5SMN1; SMN2
SCHEMBL8535813 0.72 TAS2R14 (0.36) TACR1BCHETAS2R14KCNA5PPARG
SCHEMBL7450973 0.69 ITGB1 (0.44) L3MBTL1
SCHEMBL8429207 0.69 P2RX1 (0.36) TACR1ALDH1A1L3MBTL1AKR1C3AKR1C2
SCHEMBL7450969 0.69 ITGB1 (0.44) L3MBTL1
SCHEMBL7375082 0.68 NNMT (0.34) TACR1BCHEPPARG
SCHEMBL7375079 0.68 NNMT (0.34) TACR1BCHEPPARG
SCHEMBL7376802 0.67 GPR132 (0.35) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed