SCHEMBL7376802

SCHEMBL7376802

CC(C)(C)CC(=O)N(NC(=O)c1cccc(NC=NN)c1)C(Cc1ccccc1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 1/20 0.35
SLC7A5 Q01650 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ITGB3 P05106 6/20 0.34
ITGA2B P08514 6/20 0.34
ITGB1 P05556 5/20 0.34
ITGAV P06756 5/20 0.34
ITGB5 P18084 5/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CTSL P07711 1/20 0.33
HPGDS O60760 1/20 0.33
F10 P00742 2/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7376806 1.00 GPR132 (0.35) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7380583 0.87 GPR132 (0.39) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7380590 0.87 GPR132 (0.39) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7410561 0.87 ITGB3 (0.40) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7410389 0.87 ITGB3 (0.40) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7375609 0.86 ALDH1A1 (0.39) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7375604 0.86 ALDH1A1 (0.39) GPR132SLC7A5ALDH1A1ITGB3ITGA2B
SCHEMBL7409609 0.86 ALDH1A1 (0.38) GPR132ALDH1A1CA1CA2RAB9A
SCHEMBL7409613 0.86 ALDH1A1 (0.38) GPR132ALDH1A1CA1CA2RAB9A
SCHEMBL7376793 0.85 RAB9A (0.38) ALDH1A1ITGB3ITGA2BRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed