SCHEMBL8430465

SCHEMBL8430465

CC(N[C@@H](c1ccc(F)cc1)[C@@H](O)C(=O)O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.52
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTT P42858 1/20 0.42
APAF1 O14727 1/20 0.42
ACP3 P15309 2/20 0.41
KEAP1 Q14145 2/20 0.41
NFE2L2 Q16236 2/20 0.41
MTOR P42345 1/20 0.41
POLB P06746 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8829710 1.00 NPC1 (0.52) NPC1ALDH1A1KDM4ECYP3A4CYP2D6
SCHEMBL8430344 0.91 APAF1 (0.49) ALDH1A1KDM4EAPAF1ACP3KEAP1
SCHEMBL8829781 0.91 APAF1 (0.49) ALDH1A1KDM4EAPAF1ACP3KEAP1
SCHEMBL8829775 0.85 CASR (0.48) ACP3KEAP1NFE2L2
SCHEMBL8829696 0.83 ALDH1A1 (0.48) NPC1ALDH1A1KDM4EAPAF1ACP3
SCHEMBL8430466 0.83 PHGDH (0.45) NPC1ALDH1A1CYP3A4CYP2C19APAF1
SCHEMBL8829768 0.83 PHGDH (0.45) NPC1ALDH1A1CYP3A4CYP2C19APAF1
SCHEMBL8902251 0.81 GAA (0.44) NPC1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL12154078 0.79 NPC1 (0.56) NPC1ALDH1A1KDM4ECYP3A4CYP2D6
SCHEMBL14180860 0.79 NPC1 (0.56) NPC1ALDH1A1KDM4ECYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939561-A Process for the preparation of β-phenylisoserine and β-lactam and their analogues RHONE-POULENCE RORER S.A. (FR) 1999-08-17 US disclosed
US-5763628-A Process for the preparation of β-phenylisoserine and its analogues RHONE-POULENCE RORER S.A. (FR) 1998-06-09 US disclosed