SCHEMBL8430795

SCHEMBL8430795

N=C(N)Nc1cccc(OC(=O)[C@H](Cc2ccccc2)NNC=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
LTA4H P09960 1/20 0.40
RAB9A P51151 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
LMNA P02545 1/20 0.39
IDO1 P14902 1/20 0.39
USP2 O75604 1/20 0.38
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
F10 P00742 1/20 0.38
PLAU P00749 2/20 0.37
F2 P00734 1/20 0.37
PLG P00747 1/20 0.37
PLAT P00750 1/20 0.37
KLKB1 P03952 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8432438 0.78 RAB9A (0.37) CA12CA1CA2CA9LTA4H
SCHEMBL8431230 0.77 RAB9A (0.40) CA12CA1CA2CA9LTA4H
SCHEMBL8431432 0.77 RAB9A (0.36) CA12CA1CA2CA9LTA4H
SCHEMBL8429288 0.76 CA2 (0.38) CA12CA1CA2CA9LTA4H
SCHEMBL11424081 0.76 NOS3 (0.45) CA12CA1CA2CA9LTA4H
SCHEMBL8431034 0.76 ALDH1A1 (0.41) LTA4HRAB9ALMNAUSP2PLAU
SCHEMBL8430878 0.76 CA12 (0.39) CA12CA1CA2CA9LTA4H
Hydrochloric Acid SCHEMBL11435435 0.75 NOS3 (0.44) CA12CA1CA2CA9LTA4H
Bicarbonate SCHEMBL11426039 0.75 NOS3 (0.44) CA12CA1CA2CA9LTA4H
SCHEMBL8430957 0.75 PLAU (0.38) LTA4HRAB9AUSP2PLAUF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed