SCHEMBL8433598

SCHEMBL8433598

COC(=O)c1ccc(-c2c(N)cc(C(=O)N(C(C)C)C(C)C)cc2[N+](=O)[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.46
ERN1 O75460 1/20 0.43
KMT2A Q03164 2/20 0.41
HPGD P15428 3/20 0.40
POLB P06746 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8435101 0.92 VCAM1 (0.50) VCAM1ERN1KMT2AHPGDPOLB
SCHEMBL8070684 0.88 LMNA (0.49) ERN1KMT2AMEN1SRD5A2LMNA
SCHEMBL8070686 0.88 LMNA (0.49) ERN1KMT2AMEN1SRD5A2LMNA
SCHEMBL8695884 0.87 LMNA (0.39) KMT2AHPGDPOLBCRHBPCRHR2
SCHEMBL8078533 0.79 SRD5A2 (0.51) ERN1KMT2AMEN1SRD5A2LMNA
SCHEMBL14533387 0.77 VCAM1 (0.50) VCAM1KMT2AHPGDALDH1A1MAPT
SCHEMBL8437445 0.75 SRD5A2 (0.47) ERN1KMT2AMEN1SRD5A2LMNA
SCHEMBL8437651 0.73 SRD5A2 (0.46) HPGDCA12CA1CA2CA9
SCHEMBL5434766 0.72 CA1 (0.53) KMT2AHPGDCA12CA1CA2
SCHEMBL1067197 0.72 ERN1 (0.56) VCAM1ERN1KMT2AHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965763-A Biphenyl compounds HOECHST MARION ROUSSEL (FR) 1999-10-12 US disclosed
US-5827887-A 5-ALPHA REDUCTASE INHIBITORS ROUSSEL UCLAF (FR) 1998-10-27 US disclosed