SCHEMBL8435101

SCHEMBL8435101

COC(=O)c1ccc(-c2c([N+](=O)[O-])cc(C(=O)N(C(C)C)C(C)C)cc2[N+](=O)[O-])cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.50
ERN1 O75460 1/20 0.47
KMT2A Q03164 2/20 0.44
POLB P06746 2/20 0.44
HPGD P15428 3/20 0.44
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
SRD5A2 P31213 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
LMNA P02545 1/20 0.40
AR P10275 1/20 0.40
PELP1 Q8IZL8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8433598 0.92 VCAM1 (0.46) VCAM1ERN1KMT2APOLBHPGD
SCHEMBL8078533 0.86 SRD5A2 (0.51) ERN1KMT2ASRD5A2MEN1LMNA
SCHEMBL14533387 0.81 VCAM1 (0.50) VCAM1KMT2AHPGDALDH1A1NPSR1
SCHEMBL8437445 0.80 SRD5A2 (0.47) ERN1KMT2ASRD5A2MEN1LMNA
SCHEMBL8070686 0.79 LMNA (0.49) ERN1KMT2ASRD5A2MEN1LMNA
SCHEMBL8070684 0.79 LMNA (0.49) ERN1KMT2ASRD5A2MEN1LMNA
SCHEMBL8695884 0.78 LMNA (0.39) KMT2APOLBHPGDNPSR1SRD5A2
SCHEMBL5434766 0.77 CA1 (0.53) KMT2AHPGDALDH1A1NPSR1CA12
SCHEMBL29708208 0.73 VCAM1 (0.59) VCAM1ERN1KMT2APOLBHPGD
SCHEMBL28534503 0.73 TSHR (0.62) KMT2APOLBHPGDALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965763-A Biphenyl compounds HOECHST MARION ROUSSEL (FR) 1999-10-12 US disclosed
US-5827887-A 5-ALPHA REDUCTASE INHIBITORS ROUSSEL UCLAF (FR) 1998-10-27 US disclosed