SCHEMBL8433634

SCHEMBL8433634

CC(C)[C@H](N)C(O)c1noc(C=Cc2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.36
PTGS1 P23219 1/20 0.36
ERBB2 P04626 10/20 0.36
NQO2 P16083 1/20 0.35
PDE2A O00408 1/20 0.35
CYP1A2 P05177 1/20 0.34
AHR P35869 1/20 0.33
CASP3 P42574 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8433630 1.00 TRPV1 (0.36) TRPV1PTGS1ERBB2NQO2PDE2A
Hydrochloric Acid SCHEMBL8438263 0.99 TRPV1 (0.36) TRPV1PTGS1ERBB2NQO2PDE2A
Hydrochloric Acid SCHEMBL8438272 0.99 TRPV1 (0.36) TRPV1PTGS1ERBB2NQO2PDE2A
SCHEMBL8437451 0.84 RAB9A (0.47) CYP1A2CASP3SENP8SENP7SENP6
SCHEMBL8437447 0.84 RAB9A (0.47) CYP1A2CASP3SENP8SENP7SENP6
Hydrochloric Acid SCHEMBL8433464 0.83 RAB9A (0.46) CYP1A2CASP3SENP8SENP7SENP6
SCHEMBL8433718 0.82 CASP3 (0.41) PTGS1NQO2CYP1A2AHRCASP3
SCHEMBL8433710 0.82 CASP3 (0.41) PTGS1NQO2CYP1A2AHRCASP3
Hydrochloric Acid SCHEMBL8434955 0.81 CASP3 (0.40) PTGS1NQO2CYP1A2AHRCASP3
SCHEMBL8434220 0.73 NOS3 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874585-A TREATMENT AND/OR PREVENTION OF ELASTASE-MEDIATED PROBLEMS SUCH AS ARTHRITIS, PERIODONTAL DISEASE, GLOMERULONEPHRITIS, DERMATITIS, PSORIASIS, CYSTIC FIBROSIS, CHRONIC BRONCHITIS, ALZHEIMER'S DISEASE CORTECH, INC. (US) 1999-02-23 US disclosed