SCHEMBL8434646

SCHEMBL8434646

CCOC(=O)COc1ccc(-c2cc(O)c(SCCc3ccccc3)c(=O)o2)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
HPGD P15428 4/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
TP53 P04637 2/20 0.49
HSD17B10 Q99714 2/20 0.49
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
KDM5A P29375 1/20 0.46
GAA P10253 2/20 0.43
PTPN1 P18031 1/20 0.42
EGFR P00533 10/20 0.42
GLA P06280 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6956259 0.88 XDH (0.48) HPGDALDH1A1MAPTPOLBKDM5A
SCHEMBL6952530 0.84 TNKS (0.53) KDM4EHPGDALDH1A1MAPTHSD17B10
SCHEMBL6952547 0.84 ABCB1 (0.50) MAPTCYP1A2CYP2C19PTPN1
SCHEMBL6956331 0.84 SLC16A3 (0.46) MAPT
SCHEMBL6958378 0.83 MAOA (0.45)
SCHEMBL6960907 0.83 ACHE (0.42) ALDH1A1MAPTPOLBGAA
SCHEMBL6957097 0.82 CYSLTR1 (0.41) MAPTPOLBPTPN1
SCHEMBL6963318 0.81 CYP1A1 (0.38) KDM4EHPGDALDH1A1MAPTHSD17B10
SCHEMBL6954657 0.80 SMN1; SMN2 (0.44) KDM4EHPGDALDH1A1MAPTTP53
SCHEMBL6960622 0.80 SMN1; SMN2 (0.49) KDM4EHPGDALDH1A1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed