SCHEMBL8436007

SCHEMBL8436007

Cc1cc(C(O)(C(=O)O)C(=O)O)ccc1C(C)O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 5/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C9 P11712 1/20 0.40
HIF1A Q16665 1/20 0.40
CYP1A2 P05177 3/20 0.36
GRM1 Q13255 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.34
VDR P11473 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18075239 0.74 PDE2A (0.68) PDE2A
SCHEMBL30481795 0.74 PDE2A (0.68) PDE2A
SCHEMBL8436415 0.73 HCAR3 (0.39) CYP2D6CYP2C9HIF1ACYP1A2MEN1
SCHEMBL8432092 0.73 ESR1 (0.46) CYP2D6CYP2C9HIF1ACYP1A2TDP1
SCHEMBL9156166 0.71 TDP1 (0.48) CYP2D6CYP2C9HIF1ACYP1A2TDP1
SCHEMBL25374759 0.71 PDE2A (0.50) PDE2AAR
SCHEMBL3673147 0.71 GRM1 (0.41) PDE2ACYP1A2GRM1TDP1MEN1
SCHEMBL8434483 0.70 VDR (0.49) MEN1KMT2AALDH1A1VDRAR
SCHEMBL30271542 0.69 TRPA1 (0.50) PDE2ACYP1A2TDP1ALDH1A1
SCHEMBL19205698 0.69 TRPA1 (0.50) PDE2ACYP1A2TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0605404-B1 Polycyclic dyes BASF AG (DE) 1999-12-08 EP disclosed
EP-0363034-B1 Polycyclic dyes ZENECA LTD (GB) 1995-01-04 EP disclosed
US-5212313-A For polyester IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-05-18 US disclosed
US-5183888-A Reacting a phenyl tartronic acid with a dihydrobenzofuran, oxidizing, to get dihydrobenzodifuran IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-02 US disclosed
US-5084580-A Aniline dyes for polyester fabrics to give green and blue color IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-01-28 US disclosed
EP-0363034-A2 Polycyclic dyes ZENECA LIMITED (GB) 1990-04-11 EP disclosed