SCHEMBL8438405

SCHEMBL8438405

Cc1ccc(Oc2cc(C)c(C(=O)O)cc2S(C)(=O)=O)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SLC9A1 P19634 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
HSD11B1 P28845 1/20 0.37
CSNK2A1 P68400 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439794 0.87 ALDH1A1 (0.38) ALDH1A1HPGDHSD17B10MRGPRX4HSD11B1
SCHEMBL8442180 0.85 MEN1 (0.44) HPGD
SCHEMBL8442624 0.85 MCL1 (0.45) SLC9A1
SCHEMBL8443413 0.83 SLC9A1 (0.62) SLC9A1
SCHEMBL8441138 0.82 CASP1 (0.45) ALDH1A1
SCHEMBL8059436 0.81 NR1H4 (0.46)
SCHEMBL8438984 0.81 TTR (0.51) ALDH1A1HPGDMRGPRX4
SCHEMBL8441934 0.81 BRD4 (0.47)
SCHEMBL8442155 0.80 HTT (0.56) ALDH1A1HPGD
SCHEMBL8442829 0.80 MEN1 (0.45) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708088-B1 Alkyl-5-methylsulphonyl-benzoyl-guanidine derivatives MERCK PATENT GMBH (DE) 1999-03-24 EP disclosed
US-5700839-A ANTIARRYTHMIA AGENTS; ACT AS INHIBITORS OF THE CELLULAR NA+/H+ ANTIPORTER MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-23 US disclosed
EP-0708088-A1 Alkyl-5-methylsulphonyl-benzoyl-guanidine derivatives MERCK PATENT GmbH (DE) 1996-04-24 EP disclosed