SCHEMBL8442155

SCHEMBL8442155

COc1ccccc1Oc1cc(C)c(C(=O)O)cc1S(C)(=O)=O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RAD52 P43351 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TTR P02766 1/20 0.42
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8442180 0.89 MEN1 (0.44) HTTHPGD
SCHEMBL8442829 0.86 MEN1 (0.45) HTTNPSR1KDM4EALDH1A1TTR
SCHEMBL8441897 0.86 CCR2 (0.44)
SCHEMBL8438680 0.86 CXCL8 (0.43)
SCHEMBL8059436 0.85 NR1H4 (0.46) TTR
SCHEMBL8438239 0.85 HTT (0.54) HTTLMNANPSR1KDM4EALDH1A1
SCHEMBL8438253 0.84 SLC9A1 (0.62)
SCHEMBL8439756 0.83 POLB (0.47) KDM4EALDH1A1HPGD
SCHEMBL8439161 0.83 IDO1 (0.42) ALDH1A1IDO1
SCHEMBL8441913 0.82 KDM4E (0.58) LMNAKDM4ETTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708088-B1 Alkyl-5-methylsulphonyl-benzoyl-guanidine derivatives MERCK PATENT GMBH (DE) 1999-03-24 EP disclosed
US-5700839-A ANTIARRYTHMIA AGENTS; ACT AS INHIBITORS OF THE CELLULAR NA+/H+ ANTIPORTER MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-23 US disclosed
EP-0708088-A1 Alkyl-5-methylsulphonyl-benzoyl-guanidine derivatives MERCK PATENT GmbH (DE) 1996-04-24 EP disclosed