SCHEMBL8442829

SCHEMBL8442829

COc1ccc(Oc2cc(C)c(C(=O)O)cc2S(C)(=O)=O)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TTR P02766 1/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NPC1 O15118 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439756 0.87 POLB (0.47) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL8442155 0.86 HTT (0.56) KDM4EALDH1A1TTRHTTNPSR1
SCHEMBL8441432 0.86 MEN1 (0.43) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL8441521 0.84 SLC9A1 (0.57)
SCHEMBL8441913 0.84 KDM4E (0.58) MEN1KMT2APOLBKDM4ETTR
SCHEMBL8442624 0.81 MCL1 (0.45)
SCHEMBL8438405 0.80 ALDH1A1 (0.40) ALDH1A1
SCHEMBL8059436 0.79 NR1H4 (0.46) TTR
SCHEMBL8440231 0.79 CYP1A2 (0.43)
SCHEMBL8439745 0.79 MCL1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708088-B1 Alkyl-5-methylsulphonyl-benzoyl-guanidine derivatives MERCK PATENT GMBH (DE) 1999-03-24 EP disclosed
US-5700839-A ANTIARRYTHMIA AGENTS; ACT AS INHIBITORS OF THE CELLULAR NA+/H+ ANTIPORTER MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-23 US disclosed
EP-0708088-A1 Alkyl-5-methylsulphonyl-benzoyl-guanidine derivatives MERCK PATENT GmbH (DE) 1996-04-24 EP disclosed