SCHEMBL8442192

SCHEMBL8442192

Bc1cc(OCCCCCN(C)C)cc(C(=O)OCC)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
THRB P10828 6/20 0.45
THRA P10827 6/20 0.45
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.43
ESR1 P03372 1/20 0.42
PLA2G2A P14555 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KMT2A Q03164 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
HPGD P15428 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826323 0.86 ALDH1A1 (0.53) ALDH1A1THRBTHRAKDM4EMAPT
SCHEMBL13291047 0.86 PLA2G2A (0.44) ESR1PLA2G2ACA12CA1CA2
SCHEMBL2828373 0.78 THRB (0.42) ALDH1A1THRBTHRAKDM4EMAPT
SCHEMBL27833751 0.77 ALDH1A1 (0.67) ALDH1A1THRBTHRAKDM4EMAPT
SCHEMBL5491044 0.77 PLA2G2A (0.64) ESR1PLA2G2ACA12CA1CA2
SCHEMBL9387912 0.77 PLA2G2A (0.69) ESR1PLA2G2ACA12CA1CA2
SCHEMBL20958112 0.77 PLA2G2A (0.69) ESR1PLA2G2ACA12CA1CA2
SCHEMBL2821784 0.76 ALDH1A1 (0.52) ALDH1A1KDM4EMAPTESR1KMT2A
SCHEMBL8698232 0.75 ESR1 (0.62) ALDH1A1THRBTHRAKDM4EMAPT
SCHEMBL19228932 0.73 PLA2G2A (0.59) ESR1PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed