SCHEMBL8445996

SCHEMBL8445996

CN1CCN(S(=O)(=O)c2ccc(Oc3ccc(C(=O)N=C(N)N)cc3C(F)(F)F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
SLC9A1 P19634 12/20 0.47
CYP3A4 P08684 6/20 0.47
CYP2C9 P11712 7/20 0.45
LMNA P02545 1/20 0.45
ADRA1D P25100 1/20 0.43
HTR2A P28223 1/20 0.43
SLC6A3 Q01959 1/20 0.43
SLC9A2 Q9UBY0 1/20 0.43
KMT2A Q03164 2/20 0.43
CYP2C19 P33261 4/20 0.42
KCNH2 Q12809 1/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8070565 0.99 ALDH1A1 (0.48) ALDH1A1SLC9A1CYP3A4CYP2C9LMNA
SCHEMBL8059504 0.87 ALDH1A1 (0.53) ALDH1A1CYP2C9LMNAKMT2A
SCHEMBL8445993 0.84 ALDH1A1 (0.48) ALDH1A1CYP3A4CYP2C9LMNAKMT2A
Hydrochloric Acid SCHEMBL8070562 0.83 ALDH1A1 (0.47) ALDH1A1CYP3A4CYP2C9LMNAKMT2A
SCHEMBL8070200 0.78 CCR2 (0.49) SLC9A1CYP3A4CYP2C9KMT2AKCNH2
SCHEMBL8767706 0.78 SLC9A1 (0.53) SLC9A1CYP3A4CYP2C9ADRA1DHTR2A
SCHEMBL8068662 0.77 CCR2 (0.50) SLC9A1CYP3A4CYP2C9KMT2AKCNH2
Hydrochloric Acid SCHEMBL8505886 0.77 SLC9A1 (0.52) SLC9A1CYP3A4CYP2C9ADRA1DHTR2A
Hydrochloric Acid SCHEMBL8506601 0.76 SLC9A1 (0.52) SLC9A1CYP3A4CYP2C9ADRA1DHTR2A
Hydrochloric Acid SCHEMBL8503964 0.75 SLC9A1 (0.49) SLC9A1CYP3A4CYP2C9ADRA1DHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723956-B1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AG (DE) 1999-10-13 EP claimed
EP-0723956-A1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-31 EP claimed
EP-0723956-B1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AG (DE) 1999-10-13 EP disclosed
EP-0723956-A1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-31 EP disclosed