Immethridine

Immethridine

SCHEMBL845141

c1cc(Cc2c[nH]cn2)ccn1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.44
HRH3 Q9Y5N1 3/20 0.44
CYP3A4 P08684 4/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP11B1 P15538 6/20 0.37
CYP11B2 P19099 6/20 0.37
CYP17A1 P05093 5/20 0.37
CYP19A1 P11511 3/20 0.37
LOXL2 Q9Y4K0 2/20 0.37
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
POLB P06746 1/20 0.35
LTA4H P09960 2/20 0.35
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Immethridine SCHEMBL27875904 0.90 HDAC1 (0.38) HRH4HRH3CYP3A4MAPTSMN1; SMN2
SCHEMBL649075 0.82 ALDH1A1 (0.46) HRH4HRH3SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL6973867 0.79 HDAC1 (0.37) CYP3A4SMN1; SMN2ALDH1A1CYP1A2CYP2D6
SCHEMBL6973872 0.79 GRIN2B (0.40) CYP17A1HDAC1HDAC6
SCHEMBL6972732 0.78 NOTUM (0.39) ALDH1A1CYP1A2POLBLTA4H
SCHEMBL3149298 0.78 L3MBTL1 (0.49) HRH3CYP3A4MAPTSMN1; SMN2CYP11B1
SCHEMBL6971279 0.78 HRH3 (0.38) HRH3LOXL2
SCHEMBL11050091 0.78 LPL (0.36) HRH3MAPTSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL11047959 0.78 HSP90AB1 (0.47) ALDH1A1LTA4H
SCHEMBL8001600 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240269123-A1 MUSCLE REGENERATION PROMOTER SATO PHARMACEUTICAL CO., LTD. (JP) 2024-08-15 US disclosed
CN-111670247-B Method for preparing cancer spheroids and method for selecting colorectal cancer patients 京诊断株式会社 2024-01-05 CN disclosed
US-20210147812-A1 Method of Preparing Cancer Spheroid and Method of Selecting Colorectal Cancer Patient KYO DIAGNOSTICS K.K. (JP) 2021-05-20 US disclosed
EP-3722417-A1 CANCER SPHEROID PRODUCTION METHOD AND METHOD FOR SELECTING COLON CANCER PATIENTS Kyo Diagnostics K.K. (JP) 2020-10-14 EP disclosed
CN-111670247-A Method for preparing cancer spheroids and method for selecting colorectal cancer patients 京诊断株式会社 2020-09-15 CN disclosed
CN-102481292-A Novel pharmaceutically acceptable salts of 4- (1H-imidazol-4-ylmethyl) pyridine and their therapeutic applications BIOPROJET SOC CIV 2012-05-30 CN disclosed
CN-102481292-A Novel pharmaceutically acceptable salts of 4- (1H-imidazol-4-ylmethyl) pyridine and their therapeutic applications BIOPROJET SOC CIV 2012-05-30 CN disclosed
US-20120129892-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES BIOPROJET (FR) 2012-05-24 US disclosed
US-20120129892-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES BIOPROJET (FR) 2012-05-24 US disclosed
US-20120129892-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES BIOPROJET (FR) 2012-05-24 US disclosed
EP-2432469-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES BIOPROJET (FR) 2012-03-28 EP disclosed
EP-2263672-A1 Novel pharmaceutically acceptable salts of 4-(1H-imidazol-4-ylmethyl)pyridine and their therapeutical uses BIOPROJET (FR) 2010-12-22 EP disclosed
EP-2263672-A1 Novel pharmaceutically acceptable salts of 4-(1H-imidazol-4-ylmethyl)pyridine and their therapeutical uses BIOPROJET (FR) 2010-12-22 EP disclosed
EP-2263672-A1 Novel pharmaceutically acceptable salts of 4-(1H-imidazol-4-ylmethyl)pyridine and their therapeutical uses BIOPROJET (FR) 2010-12-22 EP disclosed
WO-2010133598-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES BIOPROJET (FR) 2010-11-25 WO disclosed
WO-2010133598-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES BIOPROJET (FR) 2010-11-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120129892-A1 NOVEL PHARMACEUTICALLY ACCEPTABLE SALTS OF 4-(1H-IMIDAZOL-4-YLMETHYL)PYRIDINE AND THEIR THERAPEUTICAL USES DPP4, PDE8A, PDE8B HRH4 99/4885HRH3 513/4885CYP3A4 48/4885
US-20240269123-A1 MUSCLE REGENERATION PROMOTER MUSK, HRH3, HGF HRH4 7/4885HRH3 2/4885CYP3A4 4563/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.