SCHEMBL845214

SCHEMBL845214

CCC(=O)N1CC=C[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)CC)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
NAMPT P43490 1/20 0.38
RAB9A P51151 2/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ACE P12821 1/20 0.35
LMNA P02545 1/20 0.35
EPHX2 P34913 3/20 0.34
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL844741 0.94 ITGB1 (0.39) ITGB1ITGA4NAMPTRAB9APDE3B
SCHEMBL845097 0.87 NAMPT (0.39) ITGB1ITGA4NAMPTRAB9APDE3B
SCHEMBL845328 0.82 NAMPT (0.35) ITGB1ITGA4NAMPTRAB9APDE3B
SCHEMBL845099 0.82 ITGB1 (0.44) ITGB1ITGA4PDE3BPDE3AKDM4E
SCHEMBL845331 0.81 PTPN1 (0.41) NAMPTRAB9AKDM4EMEN1KMT2A
SCHEMBL845098 0.81 ITGB1 (0.43) ITGB1ITGA4RAB9APDE3BPDE3A
SCHEMBL845190 0.79 EPHX2 (0.42) ITGB1ITGA4RAB9AMEN1KMT2A
SCHEMBL845622 0.78 ITGB1 (0.42) ITGB1ITGA4NAMPTPDE3BALDH1A1
SCHEMBL845086 0.78 EPHX2 (0.40) ITGB1ITGA4RAB9AKDM4EMEN1
SCHEMBL13272437 0.78 ITGB1 (0.32) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed