SCHEMBL845622

SCHEMBL845622

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)Cc3cccnc3)cc2)cc1)[C@@H]1C=CCN1C(=O)Cc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
HRH3 Q9Y5N1 1/20 0.40
PAX8 Q06710 1/20 0.40
TBXAS1 P24557 2/20 0.40
POLB P06746 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
THRB P10828 1/20 0.37
NAMPT P43490 1/20 0.37
PDE3B Q13370 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845351 0.96 ITGB1 (0.41) ITGB1ITGA4HRH3PAX8TBXAS1
SCHEMBL845334 0.92 ITGB1 (0.39) ITGB1ITGA4HRH3PAX8TBXAS1
SCHEMBL872288 0.91 ITGB1 (0.37) ITGB1ITGA4HRH3PAX8TBXAS1
SCHEMBL845099 0.88 ITGB1 (0.44) ITGB1ITGA4POLBALDH1A1HTT
SCHEMBL845098 0.84 ITGB1 (0.43) ITGB1ITGA4POLBALDH1A1HTT
SCHEMBL10119337 0.82 ADRB1 (0.36) ITGB1ITGA4HRH3PAX8CHRNA7
SCHEMBL845190 0.81 EPHX2 (0.42) ITGB1ITGA4HTR1ADRD2PARP1
SCHEMBL873383 0.80 CHRNA7 (0.36) CHRNA7ALDH1A1HTTTHRBNAMPT
SCHEMBL872553 0.79 ITGB1 (0.39) ITGB1ITGA4POLBALDH1A1HTT
SCHEMBL13272435 0.79 NAPRT (0.47) ALDH1A1NAPRTTNKSPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
EP-1893573-B1 INHIBITORS OF HCV REPLICATION BRISTOL MYERS SQUIBB CO (US) 2010-07-21 EP disclosed