SCHEMBL845099

SCHEMBL845099

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)Cc3ccncc3)cc2)cc1)[C@@H]1C=CCN1C(=O)Cc1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.44
ITGA4 P13612 1/20 0.44
GLA P06280 1/20 0.42
HDAC1 Q13547 1/20 0.38
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 5/20 0.37
LMNA P02545 4/20 0.37
POLB P06746 2/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HTT P42858 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
F10 P00742 1/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845098 0.96 ITGB1 (0.43) ITGB1ITGA4GLAHDAC1TSHR
SCHEMBL872553 0.91 ITGB1 (0.39) ITGB1ITGA4GLAHDAC1TSHR
SCHEMBL845622 0.88 ITGB1 (0.42) ITGB1ITGA4POLBALDH1A1HTT
SCHEMBL845351 0.84 ITGB1 (0.41) ITGB1ITGA4POLBKMT2AALDH1A1
SCHEMBL845190 0.82 EPHX2 (0.42) ITGB1ITGA4KMT2ACA1CA2
SCHEMBL845214 0.82 ITGB1 (0.39) ITGB1ITGA4LMNAKMT2AALDH1A1
SCHEMBL845334 0.81 ITGB1 (0.39) ITGB1ITGA4HDAC1POLBKMT2A
SCHEMBL872288 0.80 ITGB1 (0.37) ITGB1ITGA4POLBPDE3B
SCHEMBL845086 0.79 EPHX2 (0.40) ITGB1ITGA4SMN1; SMN2KMT2AALDH1A1
SCHEMBL845097 0.79 NAMPT (0.39) ITGB1ITGA4SMN1; SMN2LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed