SCHEMBL845257

SCHEMBL845257

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)c3ccccc3F)cc2)cc1)[C@@H]1CCCN1C(=O)c1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.48
ALDH1A1 P00352 4/20 0.48
TSHR P16473 1/20 0.48
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
RHOC P08134 1/20 0.47
RHOA P61586 1/20 0.47
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
MAPT P10636 1/20 0.45
PABPC1 P11940 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874056 0.91 TRPV1 (0.42) TRPV1ALDH1A1TSHRCYP2C9CYP2C19
SCHEMBL845008 0.88 ALDH1A1 (0.54) ALDH1A1TSHRCYP2C9CYP2C19MEN1
SCHEMBL845343 0.87 KMT2A (0.50) TRPV1ALDH1A1TSHRMEN1KMT2A
SCHEMBL844996 0.87 CYP2C9 (0.50) TRPV1ALDH1A1CYP2C9CYP2C19MEN1
SCHEMBL845443 0.87 CYP2C9 (0.47) TRPV1ALDH1A1CYP2C9CYP2C19RHOC
SCHEMBL845013 0.85 CYP2C9 (0.46) TRPV1ALDH1A1CYP2C9CYP2C19RHOC
SCHEMBL845349 0.85 HCRTR1 (0.53) TRPV1ALDH1A1TSHRCYP2C9CYP2C19
SCHEMBL845007 0.85 PABPC1 (0.49) TRPV1ALDH1A1CYP2C9CYP2C19MEN1
SCHEMBL845458 0.85 CYP2C9 (0.46) TRPV1ALDH1A1CYP2C9CYP2C19RHOC
SCHEMBL845131 0.85 PABPC1 (0.49) TRPV1ALDH1A1CYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed