SCHEMBL8452946

SCHEMBL8452946

NN(C(=O)CCl)C(=O)c1ccco1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
ALDH1A1 P00352 4/20 0.44
POLB P06746 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
PKM P14618 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PTPN1 P18031 1/20 0.42
HDAC3 O15379 1/20 0.41
TDP1 Q9NUW8 3/20 0.41
MEN1 O00255 2/20 0.41
RECQL P46063 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
THRB P10828 1/20 0.41
APEX1 P27695 1/20 0.41
ERCC5 P28715 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7544020 0.73 CES2 (0.46) CES2CES1ALDH1A1POLBHTT
SCHEMBL5201425 0.73 CES2 (0.54) CES2CES1ALDH1A1POLBSMN1; SMN2
SCHEMBL1180379 0.72
SCHEMBL2169988 0.72 POLB (0.55) CES2CES1ALDH1A1POLBSMN1; SMN2
SCHEMBL8456803 0.72 ALDH1A1 (0.50) CES2CES1ALDH1A1POLBSMN1; SMN2
SCHEMBL9492815 0.71 HTT (0.43) CES2CES1ALDH1A1POLBSMN1; SMN2
SCHEMBL27345912 0.71 HDAC3 (0.49) CES2CES1ALDH1A1POLBSMN1; SMN2
SCHEMBL8458100 0.70 NPC1 (0.51) CES2CES1ALDH1A1POLBSMN1; SMN2
SCHEMBL28167448 0.70 CES2 (0.50) CES2CES1ALDH1A1POLBHTT
SCHEMBL10849808 0.70 CES2 (0.46) CES2CES1POLBSMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0914319-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1999-05-12 EP disclosed
WO-1997044329-A9 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS 1998-03-12 WO disclosed
WO-1997044329-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1997-11-27 WO disclosed