SCHEMBL8458100

SCHEMBL8458100

NN(C(=O)CCl)C(=O)Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
ALDH1A1 P00352 4/20 0.50
HTT P42858 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
PAX8 Q06710 2/20 0.50
GLA P06280 1/20 0.50
POLB P06746 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
AKR1B1 P15121 1/20 0.47
REN P00797 2/20 0.46
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.41
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11321849 0.82 CES1 (0.52) KMT2AMEN1ALDH1A1CES2CES1
SCHEMBL11680944 0.81 ALOX5 (0.49) NPC1RAB9AKMT2AMEN1CES2
SCHEMBL9061013 0.79 CES2 (0.48) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL9730640 0.77 MCL1 (0.46) KMT2AMEN1CES2CES1AKR1B1
SCHEMBL29291237 0.76 CES1 (0.54) KMT2AMEN1ALDH1A1CES2CES1
SCHEMBL27470447 0.76 MEN1 (0.48) KMT2AMEN1CES2CES1ALOX5
SCHEMBL8711613 0.76 ALOX5 (0.47) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL8456803 0.76 ALDH1A1 (0.50) NPC1RAB9AKMT2AMEN1TDP1
SCHEMBL4430452 0.75 CES2 (0.52) NPC1RAB9AKMT2AMEN1CES2
SCHEMBL9052467 0.74 TSHR (0.39) NPC1RAB9AKMT2AMEN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0914319-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1999-05-12 EP disclosed
WO-1997044329-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1997-11-27 WO disclosed