SCHEMBL8459394

SCHEMBL8459394

CC(CCC(=O)O)(C(=O)O)P(=O)(O)Cc1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 2/20 0.39
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP19A1 P11511 1/20 0.36
FFAR1 O14842 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ESR1 P03372 1/20 0.35
CYP3A4 P08684 1/20 0.35
ESR2 Q92731 1/20 0.35
BCHE P06276 1/20 0.35
RAB9A P51151 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALPL P05186 1/20 0.34
ALPI P09923 1/20 0.34
ALPG P10696 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8457132 0.87 KEAP1 (0.41) FDPSALDH1A1FFAR1ESR1CYP3A4
SCHEMBL8154435 0.79 HDAC3 (0.44) FDPSFFAR1SMN1; SMN2
SCHEMBL8457120 0.77 ALDH1A1 (0.44) FDPSTSHRALDH1A1RAB9ACYP1A2
SCHEMBL8159047 0.77 MAPT (0.46) SMN1; SMN2
SCHEMBL3380418 0.72 HDAC3 (0.50) FDPSTSHRFFAR1SMN1; SMN2
SCHEMBL3380551 0.72 ALDH1A1 (0.41) TSHRALDH1A1FFAR1MEN1KMT2A
SCHEMBL8585562 0.72 NAALAD2 (0.40) TSHRALDH1A1MEN1KMT2AESR1
SCHEMBL3382276 0.71 MAPT (0.50) FDPSTSHRFFAR1SMN1; SMN2
SCHEMBL8460189 0.71 ALDH1A1 (0.40) FDPSTSHRALDH1A1MEN1KMT2A
SCHEMBL7111437 0.69 NAALAD2 (0.44) FDPSTSHRALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880112-A PHOSPHINIC ACID DERIVATIVES; PROSTATE CANCER TREATMENT GUILFORD PHARMACEUTICALS INC. (US) 1999-03-09 US disclosed
US-5804602-A N-ACETYLATED ALPHA-LINKED ACIDIC DIPEPTIDASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1998-09-08 US disclosed
US-5672592-A HYDROLASE INHIBITORS, ANTITUMOR AND ANTICARCINOGENIC AGENTS, FOR PROSTATE CANCER GUILFORD PHARMACEUTICALS INC. (US) 1997-09-30 US disclosed