SCHEMBL8460189

SCHEMBL8460189

CC(CCC(=O)O)(C(=O)O)P(=O)(O)CN

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 2/20 0.40
THRB P10828 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
NAALAD2 Q9Y3Q0 1/20 0.39
ESR1 P03372 1/20 0.33
CYP3A4 P08684 1/20 0.33
ESR2 Q92731 1/20 0.33
KDM4E B2RXH2 1/20 0.31
GRM4 Q14833 1/20 0.31
FDPS P14324 1/20 0.31
TSHR P16473 3/20 0.31
GABRR1 P24046 2/20 0.31
GABRR3 A8MPY1 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
HDAC3 O15379 1/20 0.31
GABBR2 O75899 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8585562 0.83 NAALAD2 (0.40) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL3380551 0.83 ALDH1A1 (0.41) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL7111437 0.80 NAALAD2 (0.44) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL3380370 0.80 ALDH1A1 (0.39) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL3382753 0.79 NAALAD2 (0.42) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL3382732 0.77 AKR1B1 (0.39) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL8457132 0.74 KEAP1 (0.41) ALDH1A1ESR1CYP3A4ESR2FDPS
SCHEMBL3418003 0.71 NAALAD2 (0.34) ALDH1A1CYP1A2THRBKMT2AMEN1
SCHEMBL8458007 0.71 ALDH1A1 (0.35) ALDH1A1NAALAD2
SCHEMBL8459394 0.71 FDPS (0.39) ALDH1A1CYP1A2KMT2AMEN1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880112-A PHOSPHINIC ACID DERIVATIVES; PROSTATE CANCER TREATMENT GUILFORD PHARMACEUTICALS INC. (US) 1999-03-09 US disclosed
US-5804602-A N-ACETYLATED ALPHA-LINKED ACIDIC DIPEPTIDASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1998-09-08 US disclosed
US-5672592-A HYDROLASE INHIBITORS, ANTITUMOR AND ANTICARCINOGENIC AGENTS, FOR PROSTATE CANCER GUILFORD PHARMACEUTICALS INC. (US) 1997-09-30 US disclosed