SCHEMBL8460359

SCHEMBL8460359

O=C(O)Cc1cc(F)cc(CC(=O)O)c1I(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
AGBL2 Q5U5Z8 2/20 0.37
AKR1B1 P15121 2/20 0.36
AKR1A1 P14550 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CXCL8 P10145 2/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
MMP12 P39900 1/20 0.33
MMP13 P45452 1/20 0.33
MMP14 P50281 1/20 0.33
SRC P12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8460841 0.91 TSHR (0.37) TSHRAGBL2AKR1B1AKR1A1HSD17B10
SCHEMBL8464341 0.82 POLB (0.50) TSHRAKR1B1HSD17B10MEN1POLB
SCHEMBL8464321 0.80 KEAP1 (0.40) AKR1B1HSD17B10CXCL8
SCHEMBL8463501 0.80 AKR1B1 (0.36) TSHRAKR1B1HSD17B10CXCL8MEN1
SCHEMBL8459629 0.80 HPGD (0.44) TSHRAKR1B1HSD17B10MEN1POLB
SCHEMBL8462903 0.80 AKR1B1 (0.36) AKR1B1HSD17B10MEN1POLBKMT2A
SCHEMBL8460216 0.77 POLB (0.42) AKR1B1HSD17B10RXRARXRBRXRG
SCHEMBL8463402 0.77 CXCL8 (0.34) TSHRAKR1B1CXCL8MEN1KMT2A
SCHEMBL8461777 0.76 PTGS1 (0.57) TSHRAKR1B1MEN1KMT2AMMP1
SCHEMBL8464523 0.76 HSD17B10 (0.56) HSD17B10RXRARXRBRXRGPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745326-B1 Stabilization of aqueous 3-isothiazolone solutions ROHM & HAAS (US) 1999-09-22 EP disclosed
US-5594017-A WITH AN IODOSYL OR IODYL COMPOUND ROHM AND HAAS COMPANY (US) 1997-01-14 US disclosed
EP-0745326-A1 Stabilization of aqueous 3-isothiazolone solutions ROHM AND HAAS COMPANY (US) 1996-12-04 EP disclosed