SCHEMBL8460841

SCHEMBL8460841

O=C(O)Cc1cc(F)cc(F)c1I(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
CXCL8 P10145 2/20 0.36
AGBL2 Q5U5Z8 2/20 0.35
AKR1B1 P15121 2/20 0.34
AKR1A1 P14550 1/20 0.34
RIPK1 Q13546 2/20 0.33
HSD17B10 Q99714 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
PTGS1 P23219 1/20 0.32
ERN1 O75460 1/20 0.32
GPR17 Q13304 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8460359 0.91 TSHR (0.40) TSHRCXCL8AGBL2AKR1B1AKR1A1
SCHEMBL869863 0.77 RIPK1 (0.47) TSHRCXCL8AGBL2AKR1B1RIPK1
SCHEMBL29459925 0.77 RIPK1 (0.47) TSHRCXCL8AGBL2AKR1B1RIPK1
SCHEMBL8463402 0.76 CXCL8 (0.34) TSHRCXCL8AKR1B1CES2CES1
SCHEMBL20440116 0.74 AGBL2 (0.39) TSHRCXCL8AGBL2AKR1B1AKR1A1
SCHEMBL8464341 0.73 POLB (0.50) TSHRAKR1B1HSD17B10
SCHEMBL8462751 0.72 CES2 (0.45) HSD17B10CES2CES1ERN1
SCHEMBL8463501 0.72 AKR1B1 (0.36) TSHRCXCL8AKR1B1HSD17B10
SCHEMBL8464321 0.72 KEAP1 (0.40) CXCL8AKR1B1HSD17B10PTGS1
SCHEMBL8459629 0.72 HPGD (0.44) TSHRAKR1B1HSD17B10PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745326-B1 Stabilization of aqueous 3-isothiazolone solutions ROHM & HAAS (US) 1999-09-22 EP disclosed
US-5594017-A WITH AN IODOSYL OR IODYL COMPOUND ROHM AND HAAS COMPANY (US) 1997-01-14 US disclosed
EP-0745326-A1 Stabilization of aqueous 3-isothiazolone solutions ROHM AND HAAS COMPANY (US) 1996-12-04 EP disclosed