SCHEMBL8460693

SCHEMBL8460693

O=c1c2ccccc2ncn1C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.65
HTR1A P08908 1/20 0.58
HTR7 P34969 1/20 0.58
JAK2 O60674 2/20 0.55
JAK1 P23458 2/20 0.55
TYK2 P29597 2/20 0.55
JAK3 P52333 2/20 0.55
CCR5 P51681 1/20 0.51
DRD2 P14416 8/20 0.50
DRD4 P21917 7/20 0.50
DRD3 P35462 7/20 0.50
HTR6 P50406 1/20 0.48
ALDH1A1 P00352 1/20 0.48
ACVR1 Q04771 1/20 0.47
SLC6A4 P31645 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
HIF1A Q16665 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11562263 0.88 ACHE (0.54) ACHEHTR1AHTR7CCR5DRD2
SCHEMBL11567764 0.86 HTR1A (0.54) ACHEHTR1AHTR7CCR5DRD2
SCHEMBL7968829 0.83 ACHE (0.52) ACHEHTR1AHTR7JAK2JAK1
SCHEMBL17262978 0.82 ACVR1 (0.57) ACHECCR5ALDH1A1ACVR1
SCHEMBL31462149 0.82 ACVR1 (0.57) ACHECCR5ALDH1A1ACVR1
SCHEMBL31462148 0.82 ACVR1 (0.57) ACHECCR5ALDH1A1ACVR1
SCHEMBL3132276 0.82 DRD2 (0.67) ACHEJAK2JAK1TYK2JAK3
SCHEMBL11567913 0.81 ACHE (0.57) ACHEHTR1AHTR7CCR5DRD2
SCHEMBL30169432 0.80 ACVR1 (0.51) ACHECCR5DRD2ALDH1A1ACVR1
SCHEMBL11562769 0.80 CCR5 (0.47) ACHEHTR1AHTR7JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11349481-A None JP disclosed
JP-H11349481-A SIGMA RECEPTOR-BINDING AGENT EISAI CO LTD 1999-12-21 JP disclosed
US-4166117-A HYPOTENSIVES SCIENCE UNION ET CIE (FR) 1979-08-28 US disclosed