SCHEMBL8463176

SCHEMBL8463176

Cc1nc(SCCC=C(F)F)[nH]c1C

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.35
GPR84 Q9NQS5 1/20 0.34
TSHR P16473 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8462928 0.83 GPR84 (0.35) MCL1GPR84ALDH1A1POLB
SCHEMBL9045152 0.82 GPR84 (0.32) GPR84
SCHEMBL9044890 0.77 KDM4E (0.36) GPR84ALDH1A1HPGD
SCHEMBL7020173 0.74 SMN1; SMN2 (0.62) ALDH1A1HPGDPOLB
SCHEMBL8466514 0.73 GPR84 (0.31) GPR84
SCHEMBL13523375 0.69 ALDH1A1 (0.48) MCL1ALDH1A1HPGD
SCHEMBL8752059 0.69 KDM6B (0.42) ALDH1A1HPGDPOLB
SCHEMBL8752033 0.67 PKM (0.58) GPR84TSHRALDH1A1HPGDPOLB
SCHEMBL8751991 0.67 MEN1 (0.52) GPR84ALDH1A1HPGDPOLB
SCHEMBL8465490 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952359-A NEMATICIDES, INSECTICIDES AND MITICIDES; 1,1-DIFLUORO-3-(THIAZOLYL OR ISOTHIAZOYL-THIO (OR SULFINYL OR SULFONYL)-PROP-1-ENE DERIVATIVES ZENECA LIMITED (GB) 1999-09-14 US disclosed
US-5912243-A NOVEL COMPOUNDS FOR CONTROLLING NEMATODES, INSECT OR ACARID PESTS ZENECA LIMITED (GB) 1999-06-15 US disclosed
US-5705516-A NEMATOCIDES, INSECTICIDES, ACARICIDES ZENECA LIMITED (GB) 1998-01-06 US disclosed
EP-0749433-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1996-12-27 EP disclosed
WO-1995024403-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1995-09-14 WO disclosed