SCHEMBL846419

SCHEMBL846419

CCCCCN1CCCc2cc(OC(=O)Nc3cnc4ccccc4c3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.47
TRPV1 Q8NER1 8/20 0.44
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL846954 0.95 TRPV1 (0.45) ACHETRPV1KDM4ENPC1TP53
SCHEMBL846566 0.89 HSD17B10 (0.44) ACHETRPV1KDM4ENPC1TP53
SCHEMBL847501 0.86 KDM4E (0.48) ACHEKDM4ENPC1TP53RAB9A
SCHEMBL846304 0.85 TRPV1 (0.57) TRPV1KDM4ENPC1RAB9A
SCHEMBL846407 0.82 NPC1 (0.47) KDM4ENPC1TP53RAB9ASMN1; SMN2
SCHEMBL846485 0.80 HSD17B10 (0.43) TRPV1KDM4ENPC1TP53RAB9A
SCHEMBL846194 0.80 TRPV1 (0.59) TRPV1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL846869 0.79 NOTUM (0.50) KDM4ENPC1TP53RAB9ASMN1; SMN2
SCHEMBL859840 0.78 NPC1 (0.50) TRPV1KDM4ENPC1TP53RAB9A
SCHEMBL846663 0.77 TRPV1 (0.48) TRPV1RAB9AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603883-B1 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA NV (BE) 2012-03-28 EP claimed