SCHEMBL8464823

SCHEMBL8464823

O=C1C(=O)c2c(nc3cc(Cl)ccn23)-c2cccc([N+](=O)[O-])c21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 2/20 0.42
PTPRC P08575 1/20 0.39
LCK P06239 2/20 0.39
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
RECQL P46063 3/20 0.37
CA2 P00918 4/20 0.36
CA9 Q16790 4/20 0.36
CA1 P00915 3/20 0.36
CA12 O43570 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GSK3B P49841 1/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 1/20 0.36
MCL1 Q07820 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HSD11B1 P28845 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8465017 0.84 HSP90AA1 (0.56) S100A4PTPRCHSP90AA1HSP90AB1KMT2A
SCHEMBL8464968 0.83 S100A4 (0.43) S100A4PTPRCLCKIDO1TDO2
SCHEMBL8465600 0.78 HSP90AA1 (0.52) S100A4IDO1TDO2HSP90AA1HSP90AB1
SCHEMBL8466603 0.74 HSP90AA1 (0.63) S100A4PTPRCHSP90AA1HSP90AB1KMT2A
SCHEMBL8464981 0.74 HSP90AA1 (0.63) S100A4PTPRCHSP90AA1HSP90AB1KMT2A
SCHEMBL8465123 0.74 S100A4 (0.46) S100A4PTPRCLCKIDO1TDO2
SCHEMBL8465211 0.74 S100A4 (0.46) S100A4PTPRCLCKIDO1TDO2
SCHEMBL8464828 0.69 HSP90AA1 (0.61) HSP90AA1HSP90AB1
SCHEMBL9257330 0.68 S100A4 (0.77) S100A4PTPRCLCKRECQLCA2
SCHEMBL11674411 0.67 S100A4 (0.58) S100A4PTPRCLCKHSP90AA1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US disclosed