SCHEMBL8468672

SCHEMBL8468672

CCN(CC)c1cc(C)nn2c(-c3ccc(C)c(C)c3C)nnc12

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 2/20 0.39
SMPD3 Q9NY59 1/20 0.32
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5789818 0.77 CRHR1 (0.38) CRHR1SMPD3
SCHEMBL5790968 0.71 CRHR1 (0.42) CRHR1
SCHEMBL27515662 0.70 CRHR1 (0.36) CRHR1SMPD3
SCHEMBL5787555 0.69 CRHR1 (0.49) CRHR1
SCHEMBL27555107 0.63 S100B (0.36) CRHR1TP53
SCHEMBL6920917 0.61 CRHR1 (0.40) CRHR1SMPD3
SCHEMBL5789801 0.58 CRHR1 (0.44) CRHR1
SCHEMBL23854312 0.56 POLB (0.55)
SCHEMBL31673873 0.56 POLB (0.55)
SCHEMBL28930366 0.56 ALDH1A3 (0.33) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923582-A1 SUBSTITUTED 6,5-HETERO-BICYCLIC DERIVATIVES PFIZER INC. (US) 1999-06-23 EP disclosed
WO-1998008847-A1 SUBSTITUTED 6,5-HETERO-BICYCLIC DERIVATIVES PFIZER INC. (US) 1998-03-05 WO disclosed