SCHEMBL8473697

SCHEMBL8473697

CCN(CC)CC(=O)Nc1ccn(-c2ccc(N)c(Cl)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.53
SIGMAR1 Q99720 2/20 0.50
MAPT P10636 3/20 0.43
ELOVL1 Q9BW60 3/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CACNA1G O43497 1/20 0.40
CACNA1H O95180 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ENPP2 Q13822 1/20 0.38
TRPA1 O75762 1/20 0.38
LMNA P02545 1/20 0.37
AR P10275 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1356743 0.90 ABL1 (0.65) ABL1SIGMAR1MAPTELOVL1KDM4E
SCHEMBL1356441 0.78 NPC1 (0.43) ABL1SIGMAR1MAPTKDM4EALDH1A1
SCHEMBL1356872 0.77 ABL1 (0.60) ABL1SIGMAR1MAPTELOVL1KDM4E
SCHEMBL24685633 0.73 ABL1 (0.66) ABL1SIGMAR1MAPTELOVL1KDM4E
SCHEMBL1357656 0.73 ABL1 (0.73) ABL1SIGMAR1MAPTELOVL1KDM4E
SCHEMBL1356884 0.72 SIGMAR1 (0.63) ABL1SIGMAR1MAPTKDM4EALDH1A1
SCHEMBL1357515 0.72 ABL1 (0.58) ABL1SIGMAR1MAPTELOVL1KDM4E
SCHEMBL1356919 0.71 SIGMAR1 (0.52) ABL1SIGMAR1MAPTALDH1A1L3MBTL1
Oxalic Acid SCHEMBL1356980 0.70 ABL1 (0.56) ABL1SIGMAR1MAPTELOVL1KDM4E
SCHEMBL1356838 0.67 SIGMAR1 (1.00) ABL1SIGMAR1ALDH1A1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1829867-A1 Imidazole compounds having pharmaceutical activity towards the sigma receptor LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-09-05 EP disclosed