SCHEMBL8475129

SCHEMBL8475129

COC(=O)Oc1c(Cl)c(-c2ccc(Cl)cc2)oc(=O)c1-c1c(C)cc(C)cc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.39
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
TP53 P04637 3/20 0.36
CSNK2A2 P19784 2/20 0.36
CSNK2B P67870 2/20 0.36
CSNK2A1 P68400 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
APOB P04114 1/20 0.35
MTTP P55157 1/20 0.35
LMNA P02545 3/20 0.34
HSD17B10 Q99714 1/20 0.34
CETP P11597 1/20 0.33
KCNH2 Q12809 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476247 0.79 CSNK2A2 (0.46) ADORA3ALDH1A1KDM4EHPGDTP53
SCHEMBL7219386 0.74 MAPT (0.46) ADORA3ALDH1A1KDM4EHPGDTP53
SCHEMBL7223445 0.71 ADORA3 (0.37) ADORA3ALDH1A1KDM4EHPGDTP53
SCHEMBL8482317 0.67 KDM4E (0.36) ADORA3ALDH1A1KDM4EHPGDTP53
SCHEMBL9682715 0.66 RAPGEF4 (0.41) ALDH1A1KDM4EHPGDMAPTLMNA
SCHEMBL17355772 0.63 KDM4E (0.41) ALDH1A1KDM4EHPGDMAPTCYP1A2
SCHEMBL28530767 0.62 KMT2A (0.49) HPGDSMN1; SMN2
SCHEMBL19546119 0.61 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL10462265 0.60 PTGS2 (0.49) ALDH1A1TP53MAPTSMN1; SMN2LMNA
SCHEMBL14448663 0.60 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDLMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977029-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1999-11-02 US disclosed
EP-0879232-A1 3-ARYL-5-HALOGEN-PYRONE DERIVATIVES AS PEST CONTROL AGENTS BAYER AG (DE) 1998-11-25 EP disclosed
WO-1997016436-A1 3-ARYL-5-HALOGEN-PYRONE DERIVATIVES AS PEST CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-05-09 WO disclosed