SCHEMBL8475188

SCHEMBL8475188

Cc1ccc(S(=O)(=O)Nc2ccc(Oc3ccc4cc(C(=N)N)ccc4c3)c(-c3ccccc3C(=O)O)c2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44
ST14 Q9Y5Y6 1/20 0.44
PLA2G7 Q13093 3/20 0.41
POLB P06746 1/20 0.41
PARP1 P09874 1/20 0.40
PARG Q86W56 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
F2 P00734 1/20 0.40
CCR2 P41597 2/20 0.40
PKM P14618 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6295012 0.96 PLA2G7 (0.41) PRSS1PRSS2PRSS3ST14PLA2G7
SCHEMBL6300754 0.89 PRSS1 (0.47) PRSS1PRSS2PRSS3ST14PLA2G7
SCHEMBL6295817 0.88 PLA2G7 (0.46) PRSS1PRSS2PRSS3ST14PLA2G7
SCHEMBL6377229 0.86 AKR1C3 (0.52) PRSS1PRSS2PRSS3ST14POLB
Trifluoroacetic Acid SCHEMBL6294978 0.85 F2 (0.49) PRSS1PRSS2PRSS3ST14PLA2G7
SCHEMBL6295821 0.84 PLA2G7 (0.44) PRSS1PRSS2PRSS3ST14PLA2G7
SCHEMBL6300757 0.84 PLA2G7 (0.44) PRSS1PRSS2PRSS3ST14PLA2G7
Trifluoroacetic Acid SCHEMBL7154584 0.84 F2 (0.44) PRSS1PRSS2PRSS3ST14PLA2G7
Trifluoroacetic Acid SCHEMBL7158686 0.84 F2 (0.45) PRSS1PRSS2PRSS3ST14PLA2G7
Trifluoroacetic Acid SCHEMBL7157101 0.84 PLA2G7 (0.44) PRSS1PRSS2PRSS3ST14PLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1312602-A1 Amidino derivatives, and anticoagulants and thrombosis therapeutic agents containing them Eisai Co., Ltd. (JP) 2003-05-21 EP disclosed