SCHEMBL8476568

SCHEMBL8476568

Cc1ccc([C@H](CN(O)C(=O)Cc2ccc(Cl)c(Cl)c2)N2CC[C@H](O)C2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.43
OPRK1 P41145 7/20 0.41
SIGMAR1 Q99720 4/20 0.41
OPRM1 P35372 3/20 0.41
TP53 P04637 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
TSHR P16473 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TACR1 P25103 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
MTOR P42345 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
OPRD1 P41143 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550877 0.90 CCR5 (0.51) CCR5OPRK1SIGMAR1OPRM1TP53
SCHEMBL8551862 0.81 TACR1 (0.41) CCR5OPRK1OPRM1CYP2D6TACR1
SCHEMBL9098158 0.80 CCR5 (0.49) CCR5OPRK1SIGMAR1OPRM1TP53
SCHEMBL9097115 0.80 CCR5 (0.48) CCR5OPRK1SIGMAR1OPRM1TP53
SCHEMBL8553707 0.79 CCR5 (0.48) CCR5OPRK1OPRM1CYP2D6ALDH1A1
SCHEMBL9098644 0.79 CCR5 (0.47) CCR5OPRK1OPRM1TP53CYP3A4
SCHEMBL9097458 0.78 CCR5 (0.47) CCR5OPRK1SIGMAR1OPRM1TP53
SCHEMBL16333504 0.78 TACR1 (0.46) CCR5OPRK1SIGMAR1OPRM1TP53
SCHEMBL6982329 0.77 OPRK1 (0.53) CCR5OPRK1OPRM1TP53CYP3A4
SCHEMBL6982333 0.77 OPRK1 (0.53) CCR5OPRK1OPRM1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952369-A ANALGESIC, TREATMENT FOR STROKE OR ABDOMINAL PAIN ASSOCIATED WITH FUNCTIONAL BOWEL DISEASE PFIZER INC (US) 1999-09-14 US disclosed