SCHEMBL8483573

SCHEMBL8483573

Cn1cc(C(=O)NCc2ccc(O)c(O)c2)cc1C(=O)NCc1ccc(O)c(O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 8/20 0.59
ERCC4 Q92889 8/20 0.59
USP4 Q13107 1/20 0.54
USP7 Q93009 1/20 0.54
HASPIN Q8TF76 1/20 0.52
ALPG P10696 1/20 0.50
ALPL P05186 1/20 0.49
TRPV1 Q8NER1 1/20 0.45
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179001 0.79 TDP1 (0.65) POLB
SCHEMBL107157 0.78 ERCC1 (0.76) ERCC1ERCC4HASPINALPGALPL
SCHEMBL29190969 0.72 USP4 (0.61) USP4USP7HDAC3HDAC4HDAC1
SCHEMBL8269527 0.71 KDM4E (0.69) ERCC1ERCC4ALPGALPLTRPV1
SCHEMBL175299 0.70 ERCC1 (0.66) ERCC1ERCC4ALPGALPLTRPV1
SCHEMBL107288 0.70 ERCC1 (0.66) ERCC1ERCC4ALPGALPLTRPV1
SCHEMBL8506980 0.70 CA12 (0.43) POLB
SCHEMBL17231376 0.70 ALDH1A1 (0.60) ERCC1ERCC4HASPINALPGHDAC1
SCHEMBL8507242 0.69 ERCC1 (0.62) ERCC1ERCC4ALPGALPLTRPV1
SCHEMBL8507183 0.69 ERCC1 (0.62) ERCC1ERCC4ALPGALPLTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1291345-B1 Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors WARNER LAMBERT CO (US) 2005-11-30 EP disclosed