SCHEMBL29190969

SCHEMBL29190969

CC(=O)c1cc(C(=O)NCc2ccc(C#N)cc2)n(C)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP4 Q13107 1/20 0.61
USP7 Q93009 1/20 0.61
EPHX2 P34913 1/20 0.52
TP53 P04637 1/20 0.46
HDAC1 Q13547 2/20 0.45
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
KLKB1 P03952 1/20 0.45
KLK1 P06870 1/20 0.45
EGLN2 Q96KS0 2/20 0.43
KDM1A O60341 1/20 0.43
MMP2 P08253 1/20 0.43
MMP3 P08254 1/20 0.43
PPARA Q07869 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29191078 0.87 EPHX2 (0.51) USP4USP7EPHX2TP53HDAC1
SCHEMBL29191032 0.74 AKR1C3 (0.65) EPHX2HDAC1KDM1AMMP2MMP3
SCHEMBL5315293 0.72 LOXL2 (0.60) EPHX2HDAC1HDAC3HDAC2HDAC6
SCHEMBL8483573 0.72 ERCC1 (0.59) USP4USP7TP53HDAC1HDAC3
SCHEMBL27306270 0.71 USP4 (0.72) USP4USP7HDAC1HDAC3HDAC4
SCHEMBL8373038 0.71 EPHX2 (0.74) EPHX2TP53HDAC1HDAC3HDAC6
SCHEMBL12993900 0.71 EPHX2 (0.74) EPHX2TP53HDAC1KDM1AMMP2
SCHEMBL28947613 0.71 EPHX2 (0.74) EPHX2TP53HDAC1KDM1AMMP2
SCHEMBL29951484 0.70 PKM (0.47) USP4USP7HDAC8
SCHEMBL20764583 0.69 EPHX2 (0.72) EPHX2HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117886734-A Heterocyclic amide compound and preparation method, pharmaceutical composition and application thereof 中国药科大学 2024-04-16 CN disclosed