SCHEMBL8488140

SCHEMBL8488140

CCOC(=O)c1noc(C2CC2)c1C(=O)c1ccc(-n2cnnc2C)c(Br)c1C

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 14/20 0.38
GABRB3 P28472 14/20 0.38
GABRA5 P31644 14/20 0.38
GABRA1 P14867 3/20 0.33
GABRA3 P34903 3/20 0.33
GABRA2 P47869 3/20 0.33
GABRA6 Q16445 3/20 0.33
SLC22A12 Q96S37 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HCRTR2 O43614 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8488135 0.90 GABRG2 (0.36) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL8525154 0.84 HCRTR2 (0.44) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL8524136 0.83 GABRG2 (0.34) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL8525068 0.83 HCRTR2 (0.35) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL6292090 0.79 HTT (0.39) HCRTR2ALDH1A1HTT
SCHEMBL8816612 0.77 TP53 (0.41) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL8813481 0.77 HTT (0.39) HSP90AA1HCRTR2ALDH1A1HTT
SCHEMBL8525103 0.75 GABRG2 (0.35) GABRG2GABRB3GABRA5HSP90AA1HCRTR2
SCHEMBL8816565 0.75 SLC6A4 (0.39) HSP90AA1HCRTR2ALDH1A1HTT
SCHEMBL8747816 0.75 ELANE (0.42) HCRTR2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999003856-A1 4-BENZOYL-ISOXAZOLE- AND -PYRAZOLE DERIVATIVES AND 2-CYANO 1,3-DIONE DERIVATIVES AS HERBICIDES RHONE-POULENC AGRICULTURE LIMITED (GB) 1999-01-28 WO disclosed