SCHEMBL8497486

SCHEMBL8497486

CCOC(=O)CCc1cccc(C(C)NC(=O)c2cccc(NC(N)=O)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 2/20 0.42
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
ACACB O00763 1/20 0.41
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
KCNA5 P22460 2/20 0.40
KCNH2 Q12809 2/20 0.40
KCNB1 Q14721 2/20 0.40
F10 P00742 3/20 0.40
F2 P00734 2/20 0.40
KCNK2 O95069 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.39
CA2 P00918 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8499797 0.86 NAMPT (0.49) MAPTNPSR1ALDH1A1RAB9ANPC1
SCHEMBL7861961 0.82 SENP1 (0.49) MAPTALDH1A1RAB9ANPC1LMNA
SCHEMBL8497478 0.82 LMNA (0.53) MAPTALDH1A1RAB9ANPC1LMNA
SCHEMBL7377053 0.81 KMT2A (0.53) MAPTALDH1A1RAB9ANPC1LMNA
SCHEMBL7414819 0.77 HSD17B10 (0.50) MAPTNPSR1ALDH1A1RAB9ANPC1
SCHEMBL7372797 0.76 ITGB3 (0.60) MAPTRAB9ANPC1F10F2
SCHEMBL7856500 0.74 SENP1 (0.48) MAPTALDH1A1RAB9ANPC1LMNA
SCHEMBL8500098 0.74 PPARG (0.50) ALDH1A1RAB9ANPC1ACACBLMNA
SCHEMBL13091242 0.74 CYP4F2 (0.53) F10F2
SCHEMBL7348853 0.73 MAPT (0.51) MAPTALDH1A1RAB9ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed