SCHEMBL8499200

SCHEMBL8499200

CC(C)Cc1c(C(=O)N[C@H](C(=O)C(F)C(=O)C(N)CC(=O)O)C(C)C)n(C)c2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
GFER P55789 1/20 0.36
KMT2A Q03164 1/20 0.36
CASP1 P29466 1/20 0.35
CNR1 P21554 7/20 0.35
CNR2 P34972 4/20 0.35
TSHR P16473 1/20 0.35
PTGER4 P35408 6/20 0.35
EGFR P00533 2/20 0.34
OXER1 Q8TDS5 1/20 0.33
SRC P12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8496435 0.89 CASP1 (0.36) MEN1GFERKMT2ACASP1CNR1
SCHEMBL7390761 0.88 KDM4E (0.42) CASP1CNR1CNR2TSHRPTGER4
SCHEMBL7389876 0.87 PTGER4 (0.37) MEN1GFERKMT2ACNR1CNR2
SCHEMBL7200870 0.83 CASP3 (0.36) MEN1KMT2ATSHRPTGER4
SCHEMBL27564717 0.80 CNR1 (0.38) MEN1GFERKMT2ACNR1CNR2
SCHEMBL8499206 0.79 CNR1 (0.36) MEN1GFERKMT2ACNR1CNR2
SCHEMBL5670832 0.78 CASP3 (0.44) CASP1
SCHEMBL7390106 0.78 PTGER4 (0.34) MEN1KMT2ACNR1PTGER4SRC
SCHEMBL8501439 0.77 TRPA1 (0.51) MEN1KMT2ACNR2
SCHEMBL7201731 0.77 CASP3 (0.43) CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877197-A C-terminal modified (N-substituted)-2-indolyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases CONATUS PHARMACEUTICALS, INC. 1999-03-02 US disclosed