SCHEMBL8499541

SCHEMBL8499541

CC(=O)C1(c2ccccc2)C(c2ccccc2)NCCN1C([NH])=O

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CHRM1 P11229 1/20 0.33
TACR1 P25103 2/20 0.32
USP2 O75604 1/20 0.32
HHAT Q5VTY9 1/20 0.31
MEN1 O00255 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
RIPK1 Q13546 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
BRD4 O60885 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16599372 0.74 CHRM1 (0.36) POLBKDM4EALDH1A1CHRM1TACR1
SCHEMBL15094650 0.74 CHRM1 (0.36) POLBKDM4EALDH1A1CHRM1TACR1
SCHEMBL8499176 0.69 SIGMAR1 (0.36) POLBALDH1A1USP2TSHRKMT2A
SCHEMBL27749273 0.64 ALDH1A1 (0.36) KDM4EALDH1A1CHRM1TACR1MEN1
SCHEMBL5662090 0.64 OPRL1 (0.33) POLBMEN1KMT2ASLC6A2SLC6A4
SCHEMBL16599371 0.63 GAA (0.36) SLC6A2SLC6A4SLC6A3GAA
SCHEMBL11883519 0.63 SLC18A3 (0.36) POLBKDM4EALDH1A1MEN1TSHR
SCHEMBL15094674 0.62 CHRNB2 (0.36) POLBSLC6A2SLC6A4SLC6A3GAA
SCHEMBL2913724 0.61 POLB (0.42) POLBKDM4EALDH1A1MEN1TSHR
SCHEMBL16598947 0.61 GAA (0.35) ALDH1A1CHRM1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0552417-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-07 EP disclosed
EP-0528312-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-07-16 EP disclosed