SCHEMBL8500095

SCHEMBL8500095

O=C(O)CCc1cccc(CCNC(=O)c2cccc(NC(=O)NCc3ccccc3)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.59
LMNA P02545 2/20 0.55
NAMPT P43490 1/20 0.55
ROCK2 O75116 1/20 0.54
SENP1 Q9P0U3 1/20 0.52
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
RAB9A P51151 5/20 0.51
NPC1 O15118 4/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856448 0.93 PPARG (0.68) PPARGLMNASENP1HDAC2HDAC8
SCHEMBL8499211 0.87 LMNA (0.54) LMNANAMPTROCK2SENP1RAB9A
SCHEMBL7382386 0.85 PPARG (0.63) PPARGLMNANAMPTROCK2SENP1
SCHEMBL8500653 0.83 ITGB3 (0.60) PPARGLMNASENP1HDAC3HDAC4
SCHEMBL8428813 0.83 PKM (0.55) LMNANAMPTROCK2SENP1HDAC3
SCHEMBL6776908 0.82 MAPK1 (0.50) PPARGLMNASENP1HDAC2HDAC8
SCHEMBL8500098 0.81 PPARG (0.50) PPARGLMNASENP1RAB9ANPC1
SCHEMBL7372561 0.81 KCNK3 (0.56) PPARGLMNAROCK2SENP1RAB9A
SCHEMBL7014651 0.81 KDR (0.49) PPARGLMNANAMPTROCK2SENP1
SCHEMBL7380170 0.81 PPARG (0.62) PPARGLMNASENP1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed