SCHEMBL8500652

SCHEMBL8500652

N=C(N)Nc1cc(C(=O)NCc2cccc(C3(F)C=C(F)C=C(CCC(=O)O)C3)c2)cc(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
PPARG P37231 2/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
PLA2G1B P04054 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
BCHE P06276 1/20 0.36
MAPT P10636 4/20 0.36
GCGR P47871 1/20 0.36
GIPR P48546 1/20 0.36
MLYCD O95822 1/20 0.35
LMNA P02545 3/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501455 0.91 PPARG (0.43) PPARGBCHEMAPTLMNAHTT
SCHEMBL8498404 0.81 PPARG (0.43) FFAR1PPARGMAPTLMNA
SCHEMBL8526327 0.74 ITGB3 (0.49) ITGB3ITGA2B
SCHEMBL7864256 0.72 MEN1 (0.41) MEN1KMT2APLA2G1BCYP1A2CYP3A4
SCHEMBL7856467 0.71 MEN1 (0.42) PPARGMEN1KMT2APLA2G1BCYP1A2
SCHEMBL6779576 0.69 RHOC (0.48) CYP1A2GAABCHELMNAHTT
SCHEMBL7856521 0.68 PPARG (0.60) PPARGKMT2ABCHEMAPTLMNA
Hydrochloric Acid SCHEMBL6775633 0.68 RHOC (0.47) CYP1A2GAABCHELMNAHTT
SCHEMBL7450519 0.67 PPARG (0.65) FFAR1PPARGKMT2ALMNARAB9A
SCHEMBL8500892 0.66 PTGDR2 (0.35) MEN1KMT2AGAAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed