SCHEMBL8501158

SCHEMBL8501158

COCCOCCOc1cccnc1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
CYP1A2 P05177 3/20 0.42
MAPT P10636 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42
ALDH1A1 P00352 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
LMNA P02545 5/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SYK P43405 1/20 0.39
AURKB Q96GD4 1/20 0.39
INCENP Q9NQS7 1/20 0.39
ATM Q13315 2/20 0.39
NPC1 O15118 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8896957 0.85 ATM (0.37) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL9847559 0.82 CYP11B1 (0.45) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL9847563 0.79 ATM (0.39) KDM4ECYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL30867783 0.77 SMN1; SMN2 (0.51) KDM4ECYP1A2MAPTCYP2C19CYP3A4
SCHEMBL7037994 0.77 SMN1; SMN2 (0.51) KDM4ECYP1A2MAPTCYP2C19CYP3A4
SCHEMBL5349206 0.77 L3MBTL1 (0.61) KDM4EMAPTALDH1A1L3MBTL1LMNA
SCHEMBL4101620 0.77 L3MBTL1 (0.61) KDM4EMAPTALDH1A1L3MBTL1LMNA
SCHEMBL16081692 0.75 KDM4E (0.42) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL9847539 0.75 KDM4E (0.34) KDM4ECYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL31703986 0.73 CCR1 (0.46) KDM4ECYP1A2MAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772616-B1 HYDROPHILIC METAL COMPLEXES ROCHE DIAGNOSTICS GMBH (DE) 1999-12-15 EP disclosed