SCHEMBL8501225

SCHEMBL8501225

C=CCC(=O)Oc1ccc(Oc2c(-c3ccc(F)cc3)ccc3cc(OC)ccc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.43
ESR2 Q92731 8/20 0.43
GRM2 Q14416 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38
TUBB6 Q9BUF5 1/20 0.38
TUBB2B Q9BVA1 1/20 0.38
TUBB1 Q9H4B7 1/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501042 0.94 ESR1 (0.40) ESR1ESR2GRM2KDM4ETDP1
SCHEMBL8500327 0.90 ESR1 (0.42) ESR1ESR2KDM4EALDH1A1LMNA
SCHEMBL8497260 0.89 ESR1 (0.55) ESR1ESR2
SCHEMBL8501430 0.88 ESR1 (0.46) ESR1ESR2GRM2TUBB4ATUBB
SCHEMBL8500300 0.87 CYP1A2 (0.40) ESR1ESR2TDP1L3MBTL1GAA
SCHEMBL8498114 0.87 ESR1 (0.46) ESR1ESR2KDM4EALDH1A1MAPT
SCHEMBL8501370 0.85 L3MBTL1 (0.48) ESR1ESR2KDM4EALDH1A1MAPT
SCHEMBL8501283 0.83 ESR1 (0.52) ESR1ESR2
SCHEMBL8497579 0.81 SMN1; SMN2 (0.42) ESR1ESR2GRM2KDM4EMAPT
SCHEMBL7193782 0.80 ESR1 (0.47) ESR1ESR2GRM2TUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed