SCHEMBL8501413

SCHEMBL8501413

CCC(=O)Oc1ccc(Oc2c(-c3ccc(OC)c(F)c3)ccc3cc(OC)ccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.42
AKR1C2 P52895 2/20 0.42
ESR1 P03372 3/20 0.40
ESR2 Q92731 3/20 0.40
PRKCZ Q05513 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HSD17B1 P14061 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B2 P37059 1/20 0.38
PPARD Q03181 3/20 0.37
FFAR1 O14842 1/20 0.37
TRPA1 O75762 1/20 0.37
PPARA Q07869 2/20 0.36
GRM2 Q14416 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501430 0.88 ESR1 (0.46) AKR1C3AKR1C2ESR1ESR2GRM2
SCHEMBL8497579 0.88 SMN1; SMN2 (0.42) AKR1C3AKR1C2ESR1ESR2CYP1A2
SCHEMBL8497439 0.85 ESR1 (0.49) AKR1C3AKR1C2ESR1ESR2MTNR1A
SCHEMBL8502205 0.85 MTNR1A (0.43) AKR1C3AKR1C2ESR1ESR2CYP1A2
SCHEMBL8501462 0.85 ESR1 (0.47) ESR1ESR2CYP3A4CYP2D6CYP2C9
SCHEMBL8501243 0.84 KDM4E (0.39) ESR1ESR2PTGS2
SCHEMBL7190395 0.83 CYP1A2 (0.42) AKR1C3AKR1C2ESR1ESR2PRKCZ
SCHEMBL7187740 0.83 FFAR1 (0.50) AKR1C3AKR1C2ESR1CYP1A2CYP3A4
SCHEMBL7928746 0.82 DHFR (0.41) ESR1ESR2CYP1A2CYP3A4CYP2D6
SCHEMBL8497702 0.82 ESR1 (0.49) ESR1ESR2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed