SCHEMBL8506397

SCHEMBL8506397

CC(C)(C)c1ccc(C(=O)N=C(N)N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.50
SLC22A2 O15244 1/20 0.50
SLC22A1 O15245 1/20 0.50
SLC22A3 O75751 1/20 0.50
PRSS1 P07477 1/20 0.49
ACR P10323 1/20 0.49
SRD5A2 P31213 1/20 0.48
TNF P01375 1/20 0.47
KLF5 Q13887 1/20 0.47
NOD1 Q9Y239 1/20 0.47
TPH1 P17752 1/20 0.47
ESRRG P62508 1/20 0.46
SLC9A1 P19634 1/20 0.45
SLC9A2 Q9UBY0 1/20 0.45
EPHX2 P34913 1/20 0.45
NR1H4 Q96RI1 1/20 0.45
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8506609 0.98 HDAC1 (0.48) HDAC1SLC22A2SLC22A1SLC22A3PRSS1
Hydrochloric Acid SCHEMBL8341387 0.84 TPH1 (0.44) TPH1SLC9A1SLC9A2
SCHEMBL8168281 0.81 SLC9A1 (0.42) SLC9A1SLC9A2
SCHEMBL5690957 0.79 HDAC1 (0.57) HDAC1SRD5A2ESRRGEPHX2NR1H4
Hydrochloric Acid SCHEMBL8505496 0.79 HTR2B (0.41) SLC9A1SLC9A2
Hydrochloric Acid SCHEMBL8505964 0.79 CES2 (0.53) PRSS1ACRSRD5A2TPH1SLC9A1
SCHEMBL4435595 0.78 TPH1 (0.51) TPH1SLC9A1SLC9A2MEN1ALDH1A1
SCHEMBL14265179 0.78 TPH1 (0.56) TPH1SLC9A1SLC9A2KMT2ANPC1
SCHEMBL284242 0.77 EPHX2 (0.66) HDAC1SRD5A2TNFKLF5NOD1
SCHEMBL14879101 0.76 HDAC1 (0.53) HDAC1SRD5A2ESRRGEPHX2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866610-A Substituted benzoylguanidines, process for their preparation, their use as a pharmaceutical as inhibitors of the cellular NA+/H+ exchange or as a diagnostic, and pharmaceutical containing them HOECHST AKTIENGESELLSCHAFT (DE) 1999-02-02 US disclosed