SCHEMBL8514539

SCHEMBL8514539

CC(C)Oc1ccc(-c2ccnc(N3CCC(=O)CC3)n2)cc1C(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.45
DKK1 O94907 3/20 0.38
LRRK2 Q5S007 1/20 0.37
PIK3CA P42336 2/20 0.36
SORD Q00796 1/20 0.36
MTOR P42345 2/20 0.36
NEK3 P51956 1/20 0.34
LIMK1 P53667 1/20 0.34
NEK5 Q6P3R8 1/20 0.34
MYLK4 Q86YV6 1/20 0.34
STK17A Q9UEE5 1/20 0.34
SUV39H2 Q9H5I1 1/20 0.34
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3R1 P27986 1/20 0.33
PIK3CB P42338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8510840 0.89 KMO (0.43) KMODKK1LRRK2PIK3CASORD
SCHEMBL8511790 0.87 ROCK2 (0.41) KMODKK1LRRK2PIK3CAMYLK4
SCHEMBL8510671 0.86 DKK1 (0.44) KMODKK1LRRK2PIK3CASORD
Hydrochloric Acid SCHEMBL8511580 0.86 ROCK2 (0.41) KMODKK1LRRK2MYLK4STK17A
Hydrochloric Acid SCHEMBL8512525 0.86 ROCK2 (0.41) KMODKK1LRRK2MYLK4STK17A
SCHEMBL8512439 0.85 DKK1 (0.56) KMODKK1PIK3CASORDMTOR
SCHEMBL8514889 0.84 KMO (0.40) KMODKK1LRRK2MTORCTSS
Hydrochloric Acid SCHEMBL8513412 0.84 DKK1 (0.55) KMODKK1PIK3CASORDMTOR
SCHEMBL8515556 0.84 MEN1 (0.40) KMODKK1LRRK2SORDSTK17A
SCHEMBL8510713 0.84 KMO (0.39) KMODKK1LRRK2PIK3CASORD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed