SCHEMBL8514889

SCHEMBL8514889

CC(C)Oc1ccc(-c2ccnc(N3CCNC(=O)C3)n2)cc1C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.40
LRRK2 Q5S007 3/20 0.40
MTOR P42345 1/20 0.36
CTSS P25774 3/20 0.36
CTSK P43235 3/20 0.36
PRKCH P24723 1/20 0.34
PRKCE Q02156 1/20 0.34
SCN9A Q15858 1/20 0.34
GAK O14976 1/20 0.34
DKK1 O94907 1/20 0.33
AAK1 Q2M2I8 2/20 0.33
AOC3 Q16853 1/20 0.33
PRKD1 Q15139 1/20 0.33
S1PR1 P21453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511790 0.87 ROCK2 (0.41) KMOLRRK2PRKCHPRKCEDKK1
Hydrochloric Acid SCHEMBL8512525 0.86 ROCK2 (0.41) KMOLRRK2PRKCHPRKCEDKK1
Hydrochloric Acid SCHEMBL8511580 0.86 ROCK2 (0.41) KMOLRRK2PRKCHPRKCEDKK1
SCHEMBL8514539 0.84 KMO (0.45) KMOLRRK2MTORCTSSCTSK
SCHEMBL8510840 0.83 KMO (0.43) KMOLRRK2MTORDKK1
SCHEMBL8510734 0.83 ZAP70 (0.41) KMOLRRK2DKK1PRKD1
SCHEMBL8510739 0.83 ZAP70 (0.41) KMOLRRK2DKK1PRKD1
SCHEMBL8514660 0.81 KMO (0.38) KMOLRRK2MTORCTSSCTSK
SCHEMBL8510671 0.81 DKK1 (0.44) KMOLRRK2MTORDKK1
SCHEMBL8514119 0.80 SYK (0.35) DKK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed