SCHEMBL8514715

SCHEMBL8514715

Cc1nc(-c2ccc3c(c2)C(C)(C)CCC3(C)C)cc(N2CCN(C(=O)O)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARA P10276 14/20 0.46
RARB P10826 13/20 0.46
KMT2A Q03164 1/20 0.46
RARG P13631 13/20 0.44
RXRA P19793 3/20 0.42
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
CYP26A1 O43174 1/20 0.37
CYP26B1 Q9NR63 1/20 0.37
PIK3CA P42336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8512735 0.86 GPR119 (0.48) RARARARBKMT2A
SCHEMBL12959456 0.83 RARB (0.59) RARARARBRARGRXRAABCB1
SCHEMBL8514041 0.82 RARB (0.46) RARARARBRARGRXRAABCB1
SCHEMBL9612709 0.81 KMT2A (0.47) RARARARBKMT2ARARG
Trifluoroacetic Acid SCHEMBL8537644 0.81 HRH4 (0.43) RARARARBKMT2ARARGRXRA
SCHEMBL2015482 0.76 RARA (0.50) RARARARBRARG
SCHEMBL8514584 0.74 RARB (0.56) RARARARBKMT2ARARGRXRA
SCHEMBL27973420 0.73 RARA (0.47) RARARARBRARG
SCHEMBL27872046 0.72 RARA (0.46) RARARARBRARG
SCHEMBL11963431 0.70 GBA1 (0.42) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed