SCHEMBL8514987

SCHEMBL8514987

CC(C)Oc1ccc(-c2ccnc(N3CCN(/C(=N/C(=O)OC(C)(C)C)NC(=O)O)CC3)n2)cc1C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.39
TBK1 Q9UHD2 1/20 0.37
ACHE P22303 1/20 0.37
AAK1 Q2M2I8 9/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CA9 Q16790 3/20 0.36
FAAH O00519 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
CA2 P00918 2/20 0.34
CHRNA7 P36544 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8514988 1.00 KMO (0.39) KMOTBK1ACHEAAK1KDM4E
SCHEMBL8515547 0.85 ACHE (0.47) KMOTBK1ACHEFAAHCHRNA7
SCHEMBL8514120 0.78 KMO (0.40) KMOKDM4EALDH1A1LMNAGAA
Hydrochloric Acid SCHEMBL8511092 0.77 KMO (0.40) KMOKDM4EALDH1A1LMNAGAA
SCHEMBL8510840 0.76 KMO (0.43) KMOKDM4EALDH1A1HPGD
SCHEMBL8515329 0.76 ACHE (0.41) KMOACHEALDH1A1HPGD
SCHEMBL8510671 0.76 DKK1 (0.44) KMO
SCHEMBL8514539 0.76 KMO (0.45) KMOKDM4EALDH1A1LMNAGAA
SCHEMBL8515223 0.75 ACHE (0.38) TBK1ACHECA9FAAHHCAR2
SCHEMBL8515226 0.75 ACHE (0.38) TBK1ACHECA9FAAHHCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed